IRetinoid eNtsha yokuChasa ukuguga—Hydroxypinacolone Retinoate (HPR)

IHydroxypinacolone Retinoate (HPR)luhlobo lwe-ester ye-asidi ye-retinoic.Ayifani ne-retinol esters, efuna ubuncinci bamanyathelo amathathu okuguqula ukufikelela kwifom esebenzayo;ngenxa yobudlelwane obusondeleyo kunye ne-retinoic acid (yi-retinoic acid ester), i-Hydroxypinacolone Retinoate (HPR) ayifuni ukuhamba ngamanyathelo afanayo okuguqulwa njengamanye ama-retinoids - sele sele i-bioavailable kwesikhumba njengoko kunjalo.

I-Hydroxypinacolone Retinoate 10%(HPR10)yenziwe yi-Hydroxypinacolone Retinoate kunye ne-Dimethyl Isosorbide.Iyi-ester ye-All-trans Retinoic Acid, eyindalo kunye ne-synthetic derivatives ye-vitamin A, ekwazi ukubophelela kwi-retinoid receptors.Ukubophelela kwe-retinoid receptors kunokuphucula ukubonakaliswa kofuzo, okuguqula ngokufanelekileyo imisebenzi ephambili yeselula.

HPR10

Iinzuzo zeHydroxypinacolone Retinoate(HPR):

•Ukwandiswa kweMveliso yeCollagen

I-Collagen yenye yeeprotheni eziqhelekileyo emzimbeni womntu.Ifunyenwe kwizicubu zethu ezidibeneyo (i-tendon, njl njl) kunye neenwele kunye nezikhonkwane.I-collagen ephelileyo kunye nokunwebeka kwesikhumba nako kunegalelo kwimibhobho emikhulu njengoko ulusu lugoba kwaye lunweba i-pore, luyenza ibonakale inkulu.Oku kunokwenzeka kungakhathaliseki uhlobo lwesikhumba, nangona ukuba uneoli eninzi yendalo inokuthi ibonakale ngakumbi.IHydroxypinacolone Retinoate (HPR)yanceda ukwandisa amanqanaba e-collagen kulusu lwabathathi-nxaxheba.

•Ukonyuka kwe-Elastin eLusuni

IHydroxypinacolone Retinoate (HPR)kwandisa elastin eluswini.Imicu ye-elastin inika ulusu lwethu ukukwazi ukolula kwaye luphinde lubuyele endaweni.Njengoko siphulukana ne-elastin ulusu lwethu luqalisa ukugruzuka nokuthotywa.Kunye ne-collagen, i-elastin igcina ulusu lwethu lugudile kwaye luthambile, nto leyo eyenza ukuba sibonakale siqinile, sincinci.

•Nciphisa Imigca Ecolekileyo kunye nemibimbi

Ukunciphisa ukubonakala kwemibimbi mhlawumbi sesona sizathu siqhelekileyo sokuba abafazi baqale ukusebenzisa i-retinoids.Ngokuqhelekileyo iqala ngemigca emihle ejikeleze amehlo ethu, kwaye siqala ukuqaphela imibimbi emikhulu ebunzi, phakathi kwamashiya, kunye nomlomo.IHydroxypinacolone Retinoate (HPR) lolona nyango luphezulu lwemibimbi.Zisebenza kakuhle kuzo zombini ukunciphisa ukubonakala kwemibimbi kunye nokuthintela emitsha.

•Fade amabala obudala

Ekwabizwa ngokuba yi-hyperpigmentation, amabala amnyama eluswini lwethu angenzeka nakweyiphi na iminyaka kodwa athande ukuxhaphaka njengoko sikhula.Ubukhulu becala zibangelwa kukugqatswa lilanga kwaye ziba mbi kakhulu ngexesha lasehlotyeni.IHydroxypinacolone Retinoate (HPR)ingasebenza kakuhle kwi-hyperpigmentation kuba uninzi lwe-retinoids lusenza.Akukho sizathu sokulindela ukuba iHydroxypinacolone Retinoate (HPR) ibe nayiphi na eyahlukileyo.

•Phucula ithoni yolusu

I-Hydroxypinacolone Retinoate (HPR) ngokwenene yenza ulusu lwethu luzive kwaye lubukeke luncinci.I-Hydroxypinacolone Retinoate (HPR) yonyusa isantya sokuguqulwa kweeseli zesikhumba, idala ithoni yesikhumba ephuculweyo.

Inzuzo yeHPR

 Isebenza njani iHydroxypinacolone Retinoate (HPR) ngaphakathi kwesikhumba?

IHydroxypinacolone Retinoate (HPR) inokubophelela ngokuthe ngqo kwi-retinoid receptors ngaphakathi kwesikhumba nangona iyindlela ye-ester elungisiweyo ye-retinoic acid.Oku kumisela ukusabela kwekhonkco okukhokelela ekudalweni kweeseli ezintsha kubandakanywa neziyimfuneko eziya ekudaleni i-collagen kunye ne-elastin fibers.Ikwanceda ukuvuselela ukuguquka kweeseli.Uthungelwano olusisiseko lwe-collagen kunye ne-elastin fibers kunye nezinye iiseli eziyimfuneko ngaphakathi kwidermis ziba ngqindilili, zizaliswe ziiseli ezisempilweni, eziphilileyo njengesikhumba esincinci.Ikwenza oku ngokucaphuka okuncinci kunomlinganiselo olinganayo we-retinol kunye namandla angcono kunezinye ii-analog ze-Vitamin A ezifana ne-retinol esters njenge-retinyl palmitate.

 


Ixesha lokuposa: Jul-28-2023